基本的单链多肽,通过与酶的活性位点紧密结合形成复合物,抑制大多数的丝氨酸蛋白酶。
Basic single-chain polypeptide that inhibits numerous serine proteases by binding to the active site of the enzyme, forming tight complexes.
若能把抑制剂的构效关系与酶结合位点的性质联系起来研究,可能会得到更多有关除草剂抑制机理的信息。
More information about the inhibition mechanism would be gotten if the study is based on the connection of SAR of inhibitors and the property of the binding site of enzyme.
他们也设计了一个特殊的抑制物(小分子),它可以结合在人类DDAH的活性位点上。
They also designed specific inhibitors (small molecules) which bind to the active site of human DDAH.
一组称为多梳抑制复合物1(PRC1)蛋白质沉默基因必须先结合到特定的组蛋白上的甲基化位点。
A group of proteins called the polycomb repressive complex 1 (PRC1) that silences genes must first bind to a particular methylated address on a histone and.
从1945年到1955年,据两位作者估计,金融抑制使美国国债从占gdp 116%下降到了66%,整整50个百分点。
From 1945 to 1955, the authors estimate that repression reduced America's debt load by 50 percentage points, from 116% to 66% of GDP.
凝血酶及其他丝氨酸蛋白酶的不可逆抑制剂,将活性位点酰基化。比PMSF和DF P毒性小得多。
Irreversible inhibitor of Thrombin and other serine proteases. Inhibits by acylation of the active site of the enzyme. Much less toxic than PMSF and DFP.
有机酸主要通过竞争吸附位点、竞争络合等方式抑制酸性森林土壤对磷的吸附。
Organic acids inhibited adsorption of acidic forest soil to phosphorus mainly by competing adsorption sites, competitive complexing etc.
通过蛋白酶活性位点丝氨酸残基的磺酰化,不可逆的抑制丝氨酸蛋白酶。
Irreversibly inhibits serine proteases by sulfonylation of the serine residue in the active site of the protease.
可见脊髓是药物抑制伤害性信息传入的一个重要作用位点。
So we can see that the spinal cord is one of the potential target of the anesthetics inhibiting the afference of the noxious stimulation.
氧化应激可以导致DNA链断裂、DNA位点突变、DNA双链畸变和原癌基因与肿瘤抑制基因突变等形式的DNA损伤;
Oxidative stress can cause DNA damage, such as DNA strand breaks, point mutations, aberrant DNA cross-linking, and mutations in proto-oncogenes and tumor suppressor genes;
抗血小板药物通过阻断不同的作用位点抑制血小板聚集,从而达到预防及治疗血栓性疾病的作用。
They can through different sites of action blocking platelet gathered, so as to achieve the role of prevention and treatment of thrombotic disorders.
因为炎症位点的GCF中蛋白水解活性会增加,作者是否使用蛋白酶抑制剂以避免蛋白含量的降解?
Did the authors use some protease inhibitor to avoid the degradation of the protein content in the view of the increased proteolytic activity in GCF from diseased sites?
因为炎症位点的GCF中蛋白水解活性会增加,作者是否使用蛋白酶抑制剂以避免蛋白含量的降解?
Did the authors use some protease inhibitor to avoid the degradation of the protein content in the view of the increased proteolytic activity in GCF from diseased sites?
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