基本的单链多肽,通过与酶的活性位点紧密结合形成复合物,抑制大多数的丝氨酸蛋白酶。
Basic single-chain polypeptide that inhibits numerous serine proteases by binding to the active site of the enzyme, forming tight complexes.
若能把抑制剂的构效关系与酶结合位点的性质联系起来研究,可能会得到更多有关除草剂抑制机理的信息。
More information about the inhibition mechanism would be gotten if the study is based on the connection of SAR of inhibitors and the property of the binding site of enzyme.
他们也设计了一个特殊的抑制物(小分子),它可以结合在人类DDAH的活性位点上。
They also designed specific inhibitors (small molecules) which bind to the active site of human DDAH.
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