本药的化学结构类似乙酰唑胺(在氮原子上多一个甲基)。因此,药理作用及作用机制与乙酰唑胺相同。又因醋甲唑胺的结构设计减少了电离作用,故眼内透性较乙酰唑胺增强。
青光眼治疗的临床进展与研究(论著) 关键词】醋甲唑胺;乙酰唑胺;青光眼治疗;研究 [gap=532]Key words】Vinegaramine; Acetazolamide; Glaucoma treatment;Research
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... 醋甲唑胺;甲氮酰胺;甲醋唑胺;methazolamide;neptazone;neptamox;…… 甲氮酰胺 ,醋甲唑胺,甲醋唑胺;Methazolamide 酰胺;amide ...
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The drug concentration of CAP-methazolamide eye drop solutions was 400~500μg/ml, pH was 6.8~7.5.
钙纳米醋甲唑胺滴眼液的药物浓度范围400~500μg/ml,pH 6.8~7.5。
参考来源 - 钙纳米醋甲唑胺滴眼液的研制和临床前研究·2,447,543篇论文数据,部分数据来源于NoteExpress
目的探讨醋甲唑胺对青光眼的治疗价值。
Objective To study the therapeutic effect of methazolamide on glaucoma.
乙酰唑胺、醋甲唑胺、双氯非那胺等碳酸酐酶抑制剂自1954年起就被应用于青光眼的降眼压治疗。
Carbonic anhydrase inhibitors (CAIs) were first used to lower intraocular pressure (IOP) in glaucoma in 1954, with the introduction of acetazolamide, methazolamide and diclofenamide were subsequently.
结果表明,醋甲唑胺的眼用混悬剂可以显著提高药物在眼内的生物利用度,达到了局部用药制剂的设计要求。
These results indicate that the ophthalmic suspensions increased the bioavailability of MTZ in the eye aqueous humor, which is of significance in the development of topical dosage form of MTZ.
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