【正文快照】: 盐酸雷莫司琼(ramosetron hydrochloride)是一种新型高选择性5-HT3受体拮抗剂,用于治疗和预防化疗药物引起的恶心、呕吐等消化道症状。
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... 盐酸安非他酮Bupropion Hydrochloride 齐多夫定Ramosetron Hydrochloride 盐酸罗格列酮Rosiglitazone Hydrochloride ...
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Ramosetron Hydrochloride for Injection 注射用盐酸雷莫司琼 ; 注射用雷莫司琼
Ramosetron Hydrochloride Injection 盐酸雷莫司琼注射液 ; 盐酸雷莫司琼
Ramosetron Hydrochloride for Injec 注射用盐酸雷莫司琼
Ramosetron Hydrochloride for Inje 注射用盐酸雷莫司琼
Ramosetron Hydrochloride for Injiection 注射用盐酸雷莫司琼
Ramosetron Hydrochloride Orally Disintegrating Tab 盐酸雷莫司琼口内崩解片
In the synthesis process of N-methylindole,the condition of the reaction was optimized, and the yield of product was improved. The intermediate pyrrolidin-1-yl(4,5,6,7-tetra-hydro-benzo imidazol -5-yl ) methanoneand the other intermediate N-methylindole was used to produce target compound recemic ramosetron hydrochloride.
在中间体N-(4,5,6,7-四氢苯并咪唑-5基)吡咯盐酸盐和N-甲基吲哚的基础上进一步合成得到目标产物盐酸雷莫司琼。
参考来源 - 外消旋盐酸雷莫司琼的合成研究·2,447,543篇论文数据,部分数据来源于NoteExpress
Objective It's to provide reference for clinical utilization that the safety of ramosetron hydrochloride injection was studied.
目的探讨盐酸雷莫司琼注射液安全性,为临床用药提供参考。
Results Ramosetron hydrochloride injection has no hypersensitivity to guinea pig, no hemolysis and agglomeration to red blood cells of rabbit, no obvious stimulation to blood vessels of rabbit.
结果盐酸雷莫司琼注射液对豚鼠无致敏作用,对家兔红细胞无明显体外溶血及致凝集作用,对家兔血管无明显刺激作用。
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