专业释义英英释义
Partial agonist
- abstract: In pharmacology, partial agonists are drugs that bind to and activate a given receptor, but have only partial efficacy at the receptor relative to a full agonist. They may also be considered ligands which display both agonistic and antagonistic effects - when both a full agonist and partial agonist are present, the partial agonist actually acts as a competitive antagonist, competing with the full agonist for receptor occupancy and producing a net decrease in the receptor activation observed with the full agonist alone.
以上来源于: WordNet
双语例句
-
Objective:To synthesize BP897, a dopamine D3 receptor partial agonist.
前言： 目的： 合成多巴胺D， 受体部分激动剂BP897。
-
Since varenicline is only a partial agonist—not a full agonist—at the alpha4beta2 receptor site, it performs differently in smokers and nonsmokers, she said.
对alpha4beta2受体来说，既然伐伦克林仅是部分激动剂--不是完全激动剂，它对吸烟者和非吸烟者的作用是不同的，她说。
应用推荐
$firstVoiceSent
- 来自原声例句