虽然有研究表明心脏组织存在咪唑啉受体(imidazoline receptors, IR)和α2-受体,由于IR的激动剂或阻断剂同时也对α2-受体具有较高的亲和力,使得心脏IR和α2-受体的...
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胍丁胺是左旋精氨酸在左旋精氨酸脱羧酶催化下脱羧基的产物,是咪唑啉受体的内源性配体。
Agmatine formed by the decarboxylation of L-Arginine by the enzyme L-arginine decarboxylase, has been postulated to be an endogenous ligand for imidazoline receptors (I-R).
目的:在中国仓鼠卵巢(CHO)细胞上稳定转染咪唑啉1受体。
Objective: to stably transfect imidazoline-1 receptor (I 1r) in Chinese hamster ovary (CHO) cells.
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