金丝桃素有抑制中枢神经和镇静作用,用作中枢神经抑制剂和抗抑郁症。
The hypericin can inhibit nerve center and can be used as anti-depression medicine.
而且,在治疗中枢神经系统疾病方面,CB 1受体抑制剂也表现出较好的药理活性。
Furthermore, by the side of treating central nerve system disease, the antagonists of CB1 receptor show good activity too.
糖蛋白抑制剂可促进药物通过血脑屏障,对提高脑内药物的浓度和中枢神经系统药物的生物利用度具有重要意义。
P-glycoprotein inhibitors can get drugs across the blood-brain barrier. It is of great importance to improve the blood concentration in brain and bioavailability of central nervous system drugs.
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