The present invention also relates to methods of using a modulator of the GPCR.
本发明也涉及使用GPCR的调节物的方法。
So far, one third of approved small molecular drugs sold in market are the agonists or antagonists of GPCR.
目前世界药物市场上有三分之一的小分子药物是GPCR的激动剂和拮抗剂。
The unique structure and important role in the signaling transduction of GPCR make them act as very useful for drug targets.
GPCR的结构特征和在信号传导中的重要作用决定了其可以作为很好的药物靶标。
Receptor tyrosine kinases (RTK), G protein-coupled receptors (GPCR) and ion channel receptors are main cell surface receptors.
酪氨酸激酶型受体、G蛋白偶联受体和离子通道型受体是细胞表面三类主要受体。
The insect odorant receptors, as other odorant receptors from nematoid to human, have long been perceived to be G-protein-coupled receptors(GPCR).
昆虫的气味受体长久以来被认为是一种G蛋白偶联受体，遵循从线虫到人类的通用模式。
Mutant GPCR and genetic variation will cause diseases and responsible for more than 30 different human diseases which have been identified to date.
GPCR的突变及基因多态性将引发各种疾病，目前已经发现有30多种单基因疾病与此相关。
When the researchers introduced its associated membrane-impermeant fluorogen, it bound to the FAP-tagged GPCR on the cell surface, emitting a bright fluorescent glow.
当研究人员引入与其相应的膜不通透性荧光团并与细胞膜上有荧光团激活蛋白质标签的G-蛋白偶联受体结合时，发出明亮的荧光；
The present invention relates to methods of identifying whether one or more candidate compounds is a modulator of a G protein-coupled receptor (GPCR) or a modulator of blood glucose concentration.
本发明涉及鉴别一种或一种以上候选化合物是否为G蛋白偶合受体（GPCR）的调 节物或血糖浓度调节物的方法。
The present invention relates to methods of identifying whether one or more candidate compounds is a modulator of a G protein-coupled receptor (GPCR) or a modulator of blood glucose concentration.
本发明涉及鉴别一种或一种以上候选化合物是否为G蛋白偶合受体（GPCR）的调 节物或血糖浓度调节物的方法。
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