目前报道的大多数CB1拮抗剂都是利莫那班的类似物或同工物。
Most CB1 antagonists reported so far are close analogs or isosteres of rimonabant.
这些拮抗剂包括第一代抗精神病药物,如丁苯酮、吩噻嗪类药物和噻嗪类药物。
These antagonists include first generation antipsychotics such as butyrophenones, phenothiazines, and thioxanthenes.
关键是知道的性质,您的拮抗剂。
治疗冠状动脉痉挛可能涉及钙拮抗剂。
The treatment of coronary artery spasms may involve a calcium antagonist.
因此,他是轻的主要拮抗剂。
胺碘酮也可作为甲状腺激素受体拮抗剂。
Amiodarone also ACTS as a thyroid hormone receptor antagonist.
钙拮抗剂是临床常用的心血管药物之一。
Calcium antagonists is one of the commonly used cardiovascular drugs in clinic.
这是一个竞争的毒蕈碱型乙酰胆碱受体拮抗剂。
It is a competitive antagonist for the muscarinic acetylcholine receptor.
钙离子拮抗剂—尼莫地平有重要的脑保护作用。
Nimodipine, a calcium-channel antagonist has importment brain protection role.
应用组胺受体拮抗剂对防治哮喘气道重塑有一定作用。
Histamine receptor antagonists may play a role in preventing and treating airway remodeling.
因此研制和开发FGF的拮抗剂有极大的临床应用价值。
It is very important to develop antagonist of FGF for its potential of clinical use.
结论:白三烯受体拮抗剂在治疗哮喘患儿中起抗炎作用。
Conclusion: Leukotrienes receptor antagonist had anti-inflammatory effect in the treatment of asthma.
内皮素受体拮抗剂,已知对健康有益,但具体机制不明确。
Endothelin receptor antagonists are known to have health benefit but precisely why was an unknown, said Pollock, corresponding author on the study.
非竞争性拮抗剂可阻止激动剂在特定受体部位产生任何效应。
A noncompetitive antagonist prevents the agonist from producing any effect at a given receptor site.
血小板激活因子受体竞争性拮抗剂海风藤酮能抑制这种作用。
Kadsurenone which is a competitive antagonist of platelet activating factor (PAF) receptor could inhibit this effect.
目的综述新型AT 1受体拮抗剂替米沙坦的应用与研究概况。
Objective to summarize the application and research of telmisartan-new style AT1 receptor antagonists.
结论适宜浓度的烟酰胺是抗紫外线照射诱发DNA损伤的拮抗剂。
Conclusion nicotinamide is a perfect antagonist to UVR-induced DNA damage within fitting concentration.
目的观察钙拮抗剂硝苯地平对阿霉素肾病(AN)大鼠的保护作用。
Objective To investigate the protective effect of nifedipine on adriamycin nephrosis (an) and its mechanism.
前言:目的:研究钙拮抗剂尼莫地平与乌红天麻种麻的协同镇痛作用。
Objective: To study the synergism analgesic action of ges and nimodipine, a calcium antagonist.
通过计算细胞贴壁率检测BBS及其受体拮抗剂对细胞粘附能力的影响;
The effect of BBS and its receptor antagonist on cell spreading ability was detected by the percentage of cell adhesion.
静脉镁剂对心室率的影响以及心血管副作用不如钙拮抗剂或胺碘酮明显。
The effect of intravenous magnesium on the ventricular rate and its cardiovascular side effects are less significant than other calcium antagonists or amiodarone.
与阻断激动剂效应的拮抗剂不同,反向激动剂产生的效应与激动剂相反。
Different form antagonist that blocks the effect of agonist, inverse agonist produces opposite effect to that of agonist.
我们评价了卒中后早期应用血管紧张素受体拮抗剂,替米沙坦,的作用。
We evaluated the effects of therapy with an angiotensin-receptor blocker, telmisartan, initiated early after a stroke.
补充钠钾以纠正酸碱平衡,醛固酮拮抗剂和利尿剂螺内酯是主要的治疗药物。
Sodium and potassium supplements are used for the electrolyte imbalances, and aldosterone antagonists and diuretic spironolactone are mainstays of therapy.
银杏萜内酯是血小板活化因子的强拮抗剂,对心脑血管疾病具有显著的疗效。
Ginkgolides are the strong antagonists of platelet activating factors, which have notable curative effectiveness for cardio cerebrovascular diseases.
CCK受体激动剂与拮抗剂的研究深入,促进了人们对CCK生理功能的深入认识。
With study development of CCK receptor antagonist and agonist, people have deep understanding about CCK's physiological function.
结论:居主导地位的是钙拮抗剂、复方制剂以及第二代ace抑制剂——依那普利。
CONCLUSION: Calcium antagonists, compound preparations and the second generation ACE inhibitors (enalapril) are in leading position of anti-hypertensives.
因此细胞因子及其拮抗剂的研究有可能为脑缺血损伤的治疗提供一种新的思路和手段。
Study on the cytokines and their antagonists provides a new method for the therapy of cerebral ischemic injury in the future.
FDA也检查了69例牛皮癣,称皮肤病症和TNF拮抗剂之间可能存在某种的联系。
The FDA also reviewed 69 cases of psoriasis and said it found a possible link between the skin disorder and use of TNF blockers.
FDA也检查了69例牛皮癣,称皮肤病症和TNF拮抗剂之间可能存在某种的联系。
The FDA also reviewed 69 cases of psoriasis and said it found a possible link between the skin disorder and use of TNF blockers.
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