Biaryl substituted pyrazole compounds are sodium channel blockers useful for the treatment of pain and other conditions.
联芳基取代吡唑化合物为钠通道阻滞剂，用于治疗疼痛和其它病症。
Biaryl substituted pyridine, pyrimidine and pyrazine compounds are sodium channel blockers useful for the treatment of pain.
联芳基取代的吡啶、嘧啶和吡嗪化合物为用于治疗疼痛的钠通道阻滞剂。
Here we show that charged sodium-channel blockers can be targeted into nociceptors by the application of TRPV1 agonists to produce a pain-specific local anaesthesia.
结果显示，应用TRPV 1激动剂能够使带电的钠通道阻断剂特异性地作用于疼痛感受器神经元而产生特异性局麻止痛效果。
CONCLUSION Tetrandrine, as a calcium channel blockers, can reverse LVH induced by RH and elevate the cardiomyocytic membrane sodium pump and mitochondrial calcium pump activities.
结论粉防己碱因其钙拮抗作用，在降低血压、逆转左室肥厚的同时，可使细胞膜钠泵活性、线粒体钙泵活性恢复。
CONCLUSION Tetrandrine, as a calcium channel blockers, can reverse LVH induced by RH and elevate the cardiomyocytic membrane sodium pump and mitochondrial calcium pump activities.
结论粉防己碱因其钙拮抗作用，在降低血压、逆转左室肥厚的同时，可使细胞膜钠泵活性、线粒体钙泵活性恢复。
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