In the presence of hypervalent iodine reagents (PIFA), Direct coupling reaction of N-acetyl-indole with aromatic compounds provided C-3 arylated indoles in high regioselectivity.
我们使用高价有机碘试剂(PIFA)做氧化剂,实现了N-乙酰基吲哚与芳香化合物的直接偶联反应,得到了吲哚3号位高选择性的偶联产物。
In- termolecular reactions were observed with the C—Pd bond formed by the C—H activation of the aromatic ring and the nitrile group.
当然,人们也观察到了通过芳香C—H键活化产生的芳基碳钯键与腈基的分子间反应。
In- termolecular reactions were observed with the C—Pd bond formed by the C—H activation of the aromatic ring and the nitrile group.
当然,人们也观察到了通过芳香C—H键活化产生的芳基碳钯键与腈基的分子间反应。
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