Structure- activity relationship information revealed that 7-aryl-6- azaindole-1- sulfonamide derivatives was more potent than 7-anilino-6-azaindole-1- sulfonamide derivatives.
在结构与活性的关系资讯中显示， 7-苯基-6-氮基吲哚-1-磺胺类衍生物的活性比7-苯胺基-6-氮基吲哚-1-磺胺类衍 生物的活性好。
The 7-bromo group was replaced with various aniline, and then treated with 4- methoxybenzenesulfonyl chloride to afford the 6-azaindole-1-sulfonamides.
将七号位碳上的溴基取代成各种苯胺类衍生 物，再与4-甲氧基-磺基氯苯反应得到6-氮基吲哚-1-磺胺。
The 7-bromo group was replaced with various aniline, and then treated with 4- methoxybenzenesulfonyl chloride to afford the 6-azaindole-1-sulfonamides.
将七号位碳上的溴基取代成各种苯胺类衍生 物，再与4-甲氧基-磺基氯苯反应得到6-氮基吲哚-1-磺胺。
应用推荐