目的:研究具有正丁基和取代苄基侧链结构的三唑醇类化合物的抗真菌活性。
Objective:To study the antifungal activity of triazole alcohols by introducing N-butyl and substituted benzyl as side chain .
在有机合成中,芳环化合物的氯甲基化和将苄基卤氧化成芳醛或芳酮是一类极其重要的反应。
In organic synthesis, chloromethylation of aromatic compounds and oxidation of benzylic halides to aromatic aldehydes or aromatic ketones are extremely important reactions.
以化合物131为底物,对NBS/HOAC脱苄基的反应进行了研究,顺利制得脱苄基的化合物133。
Attempt to debenzylate of compound 131 with NBS/HOAC was studied and we got compound 133 having no benzyl successfully.
此外,探索通过氧化或者自由基引发,对甲苯类化合物的饱和氢活化进行苄基化反应。
Furthermore, benzylation of methyl-substituted benzene by activation of saturated hydrogen through the use of oxidation or free radical initiation has been developed.
标题化合物C24H22N2O2是由N-(4-羟基苯亚甲基)喹啉-5-胺和5,5-二甲基-1,3-环己二酮在氯化三乙基苄基铵(TEBAC)催化下以水作溶剂反应而得。
The title compound C24H22N2O2 has been synthesized by the reaction of N-arylidenenaphthalen-2-amine with 5,5-dimethyl-1,3-cyclohexadione water catalyzed by triethylbenzylammonium chlorideTEBAC.
硫酸亚铈作为一种便宜的和有效的催化剂催化芳香化合物与苄基醇、烯丙醇类化合物和苄基氯的傅-克烷基化反应。
The effects of catalyst preparation conditions and reaction parameters on the performance of the catalyst for the benzene benzylation with benzyl chloride were investigated.
本发明涉及式(I)化合物及其药用活性盐,其中R1是氢、低级烷基或苄基,其可任选地被卤素或低级烷氧基取代;
The present invention relates to compounds of formula (I) wherein R1 is hydrogen, lower alkyl or benzyl which may be optionally substituted by halogen or lower alkoxy;
合成了一系列的10-苄基吖啶酮类化合物,并探讨了一种用硼氢化钠氢化还原吖啶酮制备10-苄基-9,10-二氢吖啶的简便方法。
A series of 10-benzyl-9-acridones were synthesized and their reduction with NaBH4 to 10-benzy1-9,10-dihydroacridine derivatives was developed.
化合物3-苄基-6-氯硫色满酮的抗真茵活性与克霉唑相当。
The activity of 3-benzyl-6-chlor-thiochromanone is equal to clotrimazole's.
结果表明,经氯化汞活化的金属钐对酮类化合物与烯丙基或苄基卤代物的反应很有效,可高产率地生成叔醇。
Samarium metal (activated by HgCl2) is an effective reagent for allylation or benzylation of ketones. The corresponding tertiary alcs. are obtained in satisfactory yields.
结果表明,经氯化汞活化的金属钐对酮类化合物与烯丙基或苄基卤代物的反应很有效,可高产率地生成叔醇。
Samarium metal (activated by HgCl2) is an effective reagent for allylation or benzylation of ketones. The corresponding tertiary alcs. are obtained in satisfactory yields.
应用推荐