目的筛选桑叶中具有糖苷酶抑制活性的组分。
Objective to search for glucosidase inhibitors of various fractions extracted from Mulberry leaves.
寻求具有强xod抑制活性的天然药物及其活性成分具有重要意义。
Seeking for the natural drugs with strong XOD inhibitory activity and theirs active components is of great significance.
结论黄芩甙对我国分离的甲型流感病毒神经氨酸酶具有抑制活性的作用。
Conclusion Baicalin had inhibition effect on the strain of influenza virus isolated in China.
通过对其抑制活性的测定，证明化 合物（I）的活性很强，并且具有较好的稳定性。
The activity of the compound (I) is strong and the compound (I) has good stability which are proved by the mensuration of the inhibition activity.
本发明公开了新的具有HCV蛋白酶抑制活性的大环化合物以及制备这些化合物的方法。
The present invention discloses novel macrocyclic compounds which have HCV protease inhibitory activity as well as methods for preparing such compounds.
本论文旨在设计合成一类非核苷类对乳腺癌及HIV有抑制活性的具有潜在应用价值的新型香豆素衍生物。
This paper aims to design and synthesize a non-nucleoside class of coumarin derivatives as the lead compounds with breast cancer and HIV inhibitory activity.
本发明还公开了微生物发酵产生的对甘氨酸细胞的甘氨酸转氨酶具有抑制活性的新型的具有生理活性的物质。
Said invention also discloses a new compound with physiological activity, said new compound has inhibiting activity for glycine transferase of glycine cell and is produced by microbial fermentation.
近年来，对土茯苓化学成分及其药理作用的研究报道较多，但研究土茯苓中对酪氨酸酶有抑制活性的化合物及其抗氧化作用的报道未见。
There were a lot of reports on chemical composition and their pharmacologic action from Smilaxglabra, but studies on inhibition against tyrosinase and antioxidant activitys were not reported.
这种酶的其中一种功效是让艾滋病病毒处于关闭状态，因此一旦抑制了酶的活性，就反而会激活那些病毒基因。
One of their effects is to keep HIV genes switched off. So inhibiting their activity should switch those genes back on.
他还补充到，老鼠身上炎症状态的标志——血清淀粉减少了37%，暗示食用蔬菜可抑制炎症活性。
He added that there was a 37% reduction in serum amyloid - a marker of inflammation in mice - suggesting that vegetable consumption may inhibit inflammatory activity.
GABA通常会抑制神经活性，而且许多治疗焦虑症药物的目标就是(作用于)它的受体。
GABA typically dampens neural activity, and many drugs for treating anxiety disorders target its receptors.
异丙酚一类的药物能够作用于这类接收GABA的神经末梢，通过模拟和增强GABA引起的效果，起到抑制细胞活性的作用。
Drugs like propofol act on these GABA a receptors, mimicking and enhancing the effects of GABA, which inhibits cellular activity.
体外实验：啤酒在体外对各种酶活性均有一定程度的抑制作用。
In vitro experiment: Beer inhibited the activity of various enzymes in vitro to a certain degree.
抑制一种叫RnpA的蛋白质的活性可以终止循环，这表明Dunman的团队已经找到了关键的酶。
Blocking the activity of a protein known as RnpA stopped the recycling, indicating that Dunman's team had found a key enzyme.
这些药物通过抑制在神经肌肉接合部位水解乙酰胆碱的乙酰胆碱酯酶的活性而发挥效应。
These drugs exert their effect by inhibiting the activity of acetylcholinesterase, the enzyme that hydrolyzes acetylcholine in the neuromuscular junction.
虽然没有能够完全治愈的方法，但通过上述的方法调节水温来抑制病毒活性，可以降低死亡率，这就带来了希望。
Although there is no way to completely cure but through the above method to suppress the viral activity regulating water temperature can reduce the mortality rate which has brought hope.
治疗帕金森综合症的常用药“L - Dopa”会增加做梦的次数和活性，而抑制多巴胺的安定药会减少做梦。
L-dopa, the most popular medication for Parkinson's disease, increases the frequency and vividness of dreams, whereas antipsychotic drugs that block dopamine reduce dreaming.
一杯葡萄柚汁或吃半个葡萄柚足够抑制CYP3A4活性的一半，并且这种效应持续达24小时。
One glass of grapefruit juice, or eating half a grapefruit, is enough to suppress CYP3A4 activity by half, and the effect lasts up to 24 hours.
槟榔-正丁醇提取物对杂拟谷盗幼虫中肠淀粉酶的活性具有一定的抑制作用。
Butanolextract of areca catechu l. has certain inhibiting effect on the midgut amylase activity of confused flour beetle larvae.
在完成上述发现之后，这一研究小组又通过对大约30,000种小分子物质的检测，发现了14种物质能够抑制RnpA蛋白的活性。
Toward that end, the team screened nearly 30,000 small molecules to identify compounds that inhibit the action of RnpA.
端粒酶活性的抑制可以导致细胞的衰老和死亡。
Inhibition of telomerase activity leads the cells to senescence and death.
基本的单链多肽，通过与酶的活性位点紧密结合形成复合物，抑制大多数的丝氨酸蛋白酶。
Basic single-chain polypeptide that inhibits numerous serine proteases by binding to the active site of the enzyme, forming tight complexes.
目的：研究嵌合寡核酸对端粒酶活性的抑制作用。
Objective: To investigate the inhibitory effect of telomerase activity by chimeric oligonucleotide .
我们希望能长期的抑制成纤维细胞，同时要改善滤泡的存活性。
We hope to get chronic suppression of fibroblasts, and in that way we get improved bleb survival.
药物的精确结合能够激发或抑制特定受体的正常活性，从而在产生更有力的治疗的同时使副作用最小化。
Precise binding by a drug can stimulate or block that particular receptor's normal activity, leading to more powerful treatment while minimizing bothersome side effects.
对端粒酶活性的抑制可能是两种药物发挥抗肿瘤作用的机制之一。
The inhibition of telomerase activity may be one of the mechanisms of the anti-cancer effect of the two drugs.
对端粒酶活性的抑制可能是两种药物发挥抗肿瘤作用的机制之一。
The inhibition of telomerase activity may be one of the mechanisms of the anti-cancer effect of the two drugs.
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