雷贝拉唑(Rabeprazole)对基础胃酸和由刺激引起的胃酸分泌均有抑制作用。具体作用包括:①胃酸分泌抑制作用。②抗幽门螺杆菌作用:体外试验显示本品比奥美拉唑和兰索拉唑有更强的抗幽门螺杆菌活性,其可在几个位点直接攻击抗幽门螺杆菌,并可非竞争性、不可逆地抑制抗幽门螺杆菌的脲酶。此外,本品对胆碱受体和组胺H2受体无拮抗作用。
...;质子泵按捺剂,如埃索美拉唑(耐信),兰索拉唑(Prevacid),洛赛克(奥美拉唑),泮托拉唑(Protonix),雷贝拉唑(AcipHex)利福平(利福定,Rimactane);利福喷丁;泰利霉素(Ketek);和醋竹桃霉素(TAO)(在美国),多西紫杉醇(泰索帝)和紫杉醇(ABRA...
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世界华人消化杂志 Key Words: Rabeprazole sodium; Mosapride; Ursodeoxycholic acid; Reflux esophagitis [gap=634]关键词: 雷贝拉唑; 莫沙必利; 熊去氧胆酸; 反流性食管炎
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雷贝拉唑钠 Rabeprazole Sodium ; Sodium Rabeprazole ; AcipHex ; Rebeprazole sodium
雷贝拉唑钠肠溶片 Sodium Rabeprazole Enteric-coated Tablets ; Rabeprazole Sodium Enteric-coated Tablets ; rabeprazole sodium enteric-coated tablet ; SodiumRabepra
注射用雷贝拉唑钠 sodium rabeprazole for injetcion ; rabeprazole sodium for injection
雷贝拉唑钠肠溶胶囊 Rabeprazole Sodium Enteric-coated Capsules
雷贝拉唑杂质E Rabeprazole Sodium impurity ; Rabeprazole IMpurity
雷贝拉唑杂质A Rabeprazole Sodium impurity ; Rabeprazole Related Compound
雷贝拉唑杂质B Rabeprazole Sodium impurity ; Rabeprazole IMpurity
雷贝拉唑砜 Rabeprazole Sulfone
雷贝拉唑杂质C Rabeprazole Sodium impurity
雷贝拉唑比前期上市的其他质子泵抑制剂可以更快速的发挥作用。
Rabeprazole exerts its action much more quickly than the other proton pump inhibitors previously developed.
雷贝拉唑是一种新型的质子泵抑制剂,广泛应用于消化系统疾病的治疗。
Rabeprazole is a new type of Proton Pump Inhibitors, which is widely used in therapy for digestive system illness.
现在,让我们它快速作用的机制,关注一下雷贝拉唑是如何转化为活性形式。
Now, let's see the mechanisms for this quick action, focusing on how Rabeprazole is converted into its active form.
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