熔点:120-126℃ 相对密度:1.33g/cm3
阿折地平(Azelnidipine)是二氢吡啶类钙离子拮抗剂,用于治疗原发性高血压。阿折地平能特异性抑制血管平滑肌细胞膜电位依赖性L型钙通道,通过抑制钙离…
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阿折地平片 Azelnidipine Tablets
阿折地平中间体 Azelnidipine intermediate ; Propenoic acid,3,3-diamino-1-3-azetidinyl ester Azelnidipine intermediate ; Propenoic acid,3,3-diamino-1-3-azetidinyl ester ; Azelnidipine intermediate,2-Propenoic acid,3,3-diamino-1-3-azetidinyl ester
降血压新药阿折地平 Qilu Pharmaceutical Affairs
目的考察阿折地平的合成工艺。
本发明涉及包含由阿折地平、药用缓释材料与其它药用辅料组成的缓释制剂。
The invention relates to a slow-release preparation which comprises azelnidipine, a pharmaceutical slow-release material and other pharmaceutical auxiliary materials.
对阿折地平的合成工艺进行了研究,设计了一条适合于工业化生产的合成路线。
The synthesizing route of Azelnidipine was studied and an appropriate synthesizing process was designed for industrialization.
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