metalloproteinase inhibitor 一类组成结构中含有一个或一个以上金属离子的蛋白酶,凡能抑制此类蛋白酶又不使酶蛋白变性的物质,都属于金属蛋白酶抑制剂。 如,由田无链霉菌MD706-Y4产生的磷酰胺素(phosphoramidon),由马组链霉菌产生的塔罗肽(talopeptin)等都是金属蛋白酶抑制剂。
...,MMPs)是降解细胞外基质成分的一类重要的Zn2 依赖性蛋白水解酶,组织金属蛋白酶抑制剂(tissue inhibitor of metalloproteinases,TIMPs)是其天然抑制物,二者的表达失衡在肿瘤发生和侵袭转移过程中起着十分重要的作用。
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基质金属蛋白酶抑制剂(Tissueinhibitorofmatrixmetalloproteinases,TIMPs)是MMPs的组织抑制物,可与MMPs不可逆地结合,从而特异性抑制其活性,发挥阻止肿瘤浸润转移..
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... 硫醇蛋白酶抑制剂;thiol proteinase inhibitor 金属蛋白酶抑制剂;metalloproteinase inhibitor 酸性蛋白酶抑制剂;acid proteinase inhibitor ...
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基质金属蛋白酶抑制剂(Tissue inhibitor of matrix metalloproteinases,TIMPs)是MMPs的组织抑制物,可与MMPs不可逆地结合,从而特异性抑制其活性,发挥阻止肿瘤浸润转移 +A4...
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基质金属蛋白酶抑制剂 tissue inhibitor of metalloproteinase ; TIMP ; Matrix metallo proteinase inhibitor ; tissue inhibitor of matrix metalloproteinase
组织金属蛋白酶抑制剂 tissue inhibitor of metalloproteinase ; TIMP ; tissue inhibitor of matrix metalloproteinase
及金属蛋白酶抑制剂 TIMP ; Tissue inhibitor of metalloproteinase
金属蛋白酶组织抑制剂 TIMP ; tissue inhibitors of metalloproteinase ; tissue inhibitor of matrix metalloproteinase ; Tissue inhibitor of metalloproteinase TIMPs
和金属蛋白酶抑制剂 Tissue inhibitors of MMPs
其活性受到特异性金属蛋白酶抑制剂(TIMP)的抑制。
Their activities are inhibited by the tissue inhibitor of metalloproteinase (TIMP).
目的:评价基质金属蛋白酶抑制剂临床应用的疗效与安全性。
OBJECTIVE: to evaluate the efficiency and safety of matrix metallo-proteinase inhibitor in clinical application.
金属蛋白酶抑制剂,含有它们的药物组合物和其药物用途,其制备方法和中间体。
Inhibitors of metalloproteinase, pharmaceutical compositions containing them, their pharmaceutical application and methods and intermediate compounds for their preparation.
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