维拉帕米,一种罂粟碱的衍生物,在1962年被当作冠脉扩张剂。维拉帕米又名异搏定、戊脉安,为钙通道阻滞剂。近年来用于治疗高血压、心绞痛、心律失常、脑血管病、手指血管痉挛、腹痛、食道失驰缓症、偏头痛、肺动脉高压和预防早产。
(1)硝苯吡啶(Nifedipine)、维拉帕米(Verapamil)及硫氮卓酮(Dilthiazem):由于钙通道阻滞剂抑制钙的内流,使平滑肌收缩性下降,能降低肠易激综合征患者餐后结肠锋电位活动,有...
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...关键词】 卵巢癌细胞株;阿霉素;维拉帕米;三苯氧胺;多药耐药 [gap=1036]Key words: ovarian carcinoma cell line; adraimycin; verapamil; tamoxifen; multidrug resistance ...
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盐酸维拉帕米 Verapamil Hydrochloride ; Verapamil HCl ; VerapamilHClCAS ; Verapamil Hydrochloride Sustained-Release Tablets
盐酸维拉帕米片 Verapamil Hydrochloride Tablets
盐酸维拉帕米缓释片 Verapamil Hydrochloride Sustained-release Tablets ; Verapamil Hydrochloride Delayed-release Tablets ; Isoptin
盐酸维拉帕米注射液 Verapamil Hydrochloride Injection ; Verapamil Hydrochloride Tablets ; Verapamil Hydrochloride Inj
右维拉帕米 Dexverapamil
盐酸维拉帕米缓释胶囊 Verapamil Hydrochloride Sustained-release Capsules
维拉帕米盐酸盐 Verapamil Hydrochloride
维拉帕米.异搏定 verapamil
盐酸去甲维拉帕米 NORVERAPAMIL HYDROCHLORIDE ; Norverapamil-d7 HCl ; Norverapamil HCl
The inhibitors, cyclosporine A and verapamil,significantly enhanced the uptake amount of 9-nitrocamptothecin (. P<0.05) .
P-糖蛋白抑制剂维拉帕米能显著增加各段小肠对9-NC的吸收(P<0.05),在小肠下端更加明显。
参考来源 - 9MDR results showed that compounds 7 and 10 exhibited moderate reversal activities,and were slightly less potent than those of verapamil against K562 cell line. It is believed that compounds 7 and 10 have MDR activity.
结果和结论:化合物的结构均由核磁共振氢谱,质谱,红外和元素分析确证,活性实验结果显示,化合物7,10逆转活性略低于维拉帕米,但是仍具有一定的多药耐药逆转活性。
参考来源 - 1·2,447,543篇论文数据,部分数据来源于NoteExpress
结论:维拉帕米可增强细辛水煎剂的镇痛作用。
CONCLUSION: Verapamil can enhance the analgesic action of Asarum water decoction.
目的观察维拉帕米联合利多卡因对兔表面麻醉作用的影响。
Objective To observe the surface anesthetic effect of verapamil hydrochloride combined with lidocaine hydrochloride on rabbits.
我们推断糖尿病弱氟卡胺、 E-4031和维拉帕米的心律失常作用。
We concluded that diabetes mellitus reduces the antiarrhythmic effects of flecainide , E-4031, and verapamil.
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