乙哌立松(Eperisone)为中枢性肌肉松弛药。作用于脊髓和血管平滑肌,通过抑制脊髓反射,抑制γ-运动神经元的自发性冲动,减轻肌梭的灵敏度,从而缓解骨骼肌的紧张;并通过扩张血管而改善血液循环,从多方面阻断肌紧张亢进→循环障碍→肌疼痛→肌紧张亢进这种骨骼肌紧张的恶性循环。
(5)乙哌立松(eperisone):乙哌立松属骨骼肌松弛药,除可抑制肌张力过高并可抑制疼痛反射活动,从而改善紧张型头痛的症状。口服剂量150mg/d,分次服用。
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结论:方法快速、准确、专一性强,适用于盐酸乙哌立松片的含量测定。
CONCLUSION:The method was simple, sensitive, rapid and suitable for the quantitative anylysis of the preparation.
目的:验证乙哌立松对伴有颅周肌肉收缩的急性或慢性紧张型头痛的临床疗效。
AIM: To evaluate the clinical effects of eperisone in the treatment of chronic tension_type headache associated with pericranial muscle contraction.
结论盐酸乙哌立松可以改善VP患者的肌张力,能否能提高患者的日常生活才干尚有待进一步研讨。
Conclusion eperisone can improve hypermyotonia, whether eperisone can promote the daily life ability of VP patients should be study further.
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