早期、剂量、脉注射是应用盐酸纳洛酮治疗的关键。
The key of naloxone therapy is early large dose naloxone intravenous injection.
盐酸纳洛酮在动物试验和临床中早期主要应用于麻醉复苏、酒精中毒、毒品中毒、休克、昏迷及中风的治疗,并取得了良好的效果。
In animal test and clinic anesthesia resuscitation, alcoholism, drug intoxication, shock, coma and stoke were treated by naloxone, and got excellent outcomes.
但由于该药肝脏首过效应严重,口服无效,目前国内外临床上供应用的盐酸纳洛酮的剂型为注射液和舌下片。
Because of a serious liver first-pass effect, the dosage forms of Naloxone Hydrochloride is mainly used on domestic and aboard clinical practice in the forms of injection and sublingual tablet.
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